SCHEMBL8744826

SCHEMBL8744826

COc1ccc(C[C@H](NC(=O)Cc2c(C)cc(C)cc2C)C(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.54
ITGA4 P13612 1/20 0.54
FPR2 P25090 1/20 0.53
KMT2A Q03164 1/20 0.53
LDHA P00338 1/20 0.51
CA2 P00918 1/20 0.51
ALDH1A1 P00352 1/20 0.48
ALOX15 P16050 1/20 0.48
ALB P02768 1/20 0.47
IL2 P60568 1/20 0.47
PTPN1 P18031 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ITGB3 P05106 1/20 0.47
ITGAV P06756 1/20 0.47
ITGA5 P08648 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8744821 1.00 ITGB1 (0.54) ITGB1ITGA4FPR2KMT2ALDHA
SCHEMBL9594665 0.89 ALDH1A1 (0.50) ITGB1ITGA4KMT2ALDHAALDH1A1
SCHEMBL8744831 0.89 ALDH1A1 (0.50) ITGB1ITGA4KMT2ALDHAALDH1A1
SCHEMBL8744782 0.87 L3MBTL1 (0.57) ITGB1ITGA4L3MBTL1ITGB3
SCHEMBL8744788 0.87 L3MBTL1 (0.57) ITGB1ITGA4L3MBTL1ITGB3
SCHEMBL5189503 0.82 FPR2 (0.68) FPR2KMT2ALDHAALDH1A1ALOX15
SCHEMBL9790211 0.81 HTT (0.59) FPR2KMT2ALDHACA2PTPN1
SCHEMBL9790209 0.81 HTT (0.59) FPR2KMT2ALDHACA2PTPN1
SCHEMBL8744805 0.79 TACR1 (0.57) KMT2AALDH1A1L3MBTL1
SCHEMBL9594563 0.79 TACR1 (0.57) KMT2AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed