SCHEMBL8744966

SCHEMBL8744966

COc1cccc(N2CCN(Cc3ccc(CC(=O)O)cc3)CC2)c1

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.71
SMN1; SMN2 Q16637 2/20 0.71
ALDH1A1 P00352 1/20 0.71
MAPT P10636 3/20 0.65
TSHR P16473 2/20 0.65
HSD17B10 Q99714 2/20 0.64
TP53 P04637 1/20 0.64
ITGB3 P05106 4/20 0.60
ITGA2B P08514 4/20 0.60
GFER P55789 3/20 0.59
LMNA P02545 1/20 0.58
SIGMAR1 Q99720 1/20 0.58
KMT2A Q03164 2/20 0.55
KCNH2 Q12809 2/20 0.55
DRD2 P14416 1/20 0.55
MEN1 O00255 1/20 0.54
CHRM4 P08173 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8745027 0.99 KDM4E (0.70) KDM4ESMN1; SMN2ALDH1A1MAPTTSHR
SCHEMBL8744975 0.86 ITGB3 (0.64) ALDH1A1MAPTHSD17B10ITGB3ITGA2B
SCHEMBL7655244 0.85 DRD2 (0.60) KDM4ESMN1; SMN2ALDH1A1GFERKMT2A
Hydrochloric Acid SCHEMBL8745028 0.83 KDM4E (0.68) KDM4ESMN1; SMN2ALDH1A1MAPTTSHR
SCHEMBL25370948 0.83 KDM4E (0.80) KDM4ESMN1; SMN2ALDH1A1MAPTTSHR
SCHEMBL6031705 0.83 KDM4E (1.00) KDM4ESMN1; SMN2ALDH1A1MAPTTSHR
SCHEMBL27395515 0.83 KDM4E (0.80) KDM4ESMN1; SMN2ALDH1A1MAPTTSHR
SCHEMBL8691440 0.83 DRD4 (0.70) ALDH1A1MAPTITGB3ITGA2BGFER
SCHEMBL11549618 0.82 KDM4E (0.78) KDM4ESMN1; SMN2ALDH1A1MAPTTSHR
Hydrochloric Acid SCHEMBL8690310 0.82 DRD4 (0.68) ITGB3ITGA2BGFERDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0753515-A2 Benzylpiperazine derivatives as antiallergic and anti-inflammatory agents Senju Pharmaceutical Co., Ltd. (JP) 1997-01-15 EP claimed
EP-0753515-A2 Benzylpiperazine derivatives as antiallergic and anti-inflammatory agents Senju Pharmaceutical Co., Ltd. (JP) 1997-01-15 EP disclosed