SCHEMBL8745768

SCHEMBL8745768

CCOc1cc2c(C)c(CCOS(C)(=O)=O)c(=O)oc2cc1OC

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.44
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
ALDH1A2 O94788 2/20 0.42
ALDH1A1 P00352 2/20 0.42
ALDH2 P05091 2/20 0.42
ALDH1B1 P30837 2/20 0.42
ALDH1A3 P47895 2/20 0.42
POLB P06746 3/20 0.41
MAPT P10636 1/20 0.41
F11 P03951 2/20 0.40
ACHE P22303 2/20 0.40
CTSG P08311 1/20 0.40
KLK7 P49862 1/20 0.40
KLK14 Q9P0G3 1/20 0.40
KLK5 Q9Y337 1/20 0.40
STS P08842 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745784 0.93 NQO1 (0.50) NQO1ALDH1A2ALDH1A1ALDH2ALDH1B1
SCHEMBL8745814 0.83 NQO1 (0.52) NQO1PDE3BPDE3AALDH1A2ALDH1A1
SCHEMBL8807846 0.81 ACHE (0.48) NQO1PDE3BPDE3AMAPTACHE
SCHEMBL8807713 0.77 ALDH1A1 (0.48) NQO1PDE3BPDE3AALDH1A2ALDH1A1
SCHEMBL9148098 0.77 ALDH1A1 (0.48) NQO1ALDH1A2ALDH1A1ALDH2ALDH1B1
SCHEMBL8745770 0.77 ALDH1A1 (0.57) NQO1ALDH1A2ALDH1A1ALDH1B1ALDH1A3
SCHEMBL8745789 0.76 ALDH1A1 (0.55) ALDH1A1KMT2A
SCHEMBL8745792 0.76 NQO1 (0.47) NQO1ALDH1A2ALDH1A1ALDH2ALDH1B1
SCHEMBL9144825 0.76 NQO1 (0.50) NQO1ALDH1A2ALDH1A1ALDH2ALDH1B1
SCHEMBL8745793 0.75 NQO1 (0.56) NQO1ALDH1A2ALDH1A1ALDH2ALDH1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed
EP-0663911-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE. SCHWABE WILLMAR GMBH & CO (DE) 1995-07-26 EP disclosed
WO-1994008985-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1994-04-28 WO disclosed