SCHEMBL874591

SCHEMBL874591

COCCc1ccccc1[N+](=O)[O-]

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.56
TSHR P16473 1/20 0.56
TDP1 Q9NUW8 1/20 0.52
HPGD P15428 1/20 0.51
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
RECQL P46063 1/20 0.50
L3MBTL1 Q9Y468 3/20 0.48
GAA P10253 2/20 0.48
MAPT P10636 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 2/20 0.47
HSD17B10 Q99714 1/20 0.47
MAOB P27338 1/20 0.47
KMT2A Q03164 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
PTPN1 P18031 1/20 0.46
MEN1 O00255 2/20 0.46
ACHE P22303 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20749087 0.89 ALDH1A1 (0.53) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL28912669 0.88 ALDH1A1 (0.51) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL27258885 0.86 TDP1 (0.56) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL7135820 0.85 ALDH1A1 (0.60) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL261866 0.83 ALDH1A1 (0.58) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL12064619 0.82 ALDH1A1 (0.53) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL8393234 0.82 ALDH1A1 (0.53) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL3202573 0.82 ALDH1A1 (0.72) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL8957406 0.81 ALDH1A1 (0.56) ALDH1A1TSHRTDP1HPGDNPC1
SCHEMBL17339105 0.81 ALDH1A1 (0.56) ALDH1A1TSHRTDP1HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704130-A1 SYNTHESIS OF BORONATE ESTER DERIVATIVES AND USES THEREOF Melinta Therapeutics, Inc. (US) 2020-09-09 EP disclosed
EP-3615544-A1 ANTITUMORAL COMPOUNDS Pharma Mar S.A. (ES) 2020-03-04 EP disclosed
WO-2018197663-A1 ANTITUMORAL COMPOUNDS PHARMA MAR, S.A. (ES) 2018-11-01 WO disclosed
WO-2018167270-A1 ANTICANCER COMPOUNDS PHARMA MAR, S.A. (ES) 2018-09-20 WO disclosed
EP-3140310-A1 SYNTHESIS OF BORONATE SALTS AND USES THEREOF Rempex Pharmaceuticals, Inc. (US) 2017-03-15 EP disclosed
WO-2015171430-A1 SYNTHESIS OF BORONATE SALTS AND USES THEREOF REMPEX PHARMACEUTICALS, INC. (US) 2015-11-12 WO disclosed
EP-2825542-A1 LIVER X RECEPTOR MODULATORS Vitae Pharmaceuticals, Inc. (US) 2015-01-21 EP disclosed
WO-2013138568-A1 LIVER X RECEPTION MODULATORS VITAE PHARMACEUTICALS, INC. (US) 2013-09-19 WO disclosed
EP-2576569-A1 SYNTHETIC PROCESS FOR THE MANUFACTURE OF ECTEINASCIDIN COMPOUNDS Pharma Mar S.A. (ES) 2013-04-10 EP disclosed
WO-2012040242-A1 SUBSTITUTED PROLINE INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-03-29 WO disclosed
US-20030181742-A1 Process for the preparation of pregnane derivatives KURARAY CO., LTD. (JP) 2003-09-25 US disclosed
EP-1325928-A1 PROCESS FOR THE PREPARATION OF PREGNANE DERIVATIVES Kuraray Co., Ltd. (JP) 2003-07-09 EP disclosed
US-5984975-A COLORFAST, WASHFAST HAIR DYES L'OREAL (FR) 1999-11-16 US disclosed
US-5703266-A OXIDATION HAIR DYES L'OREAL (FR) 1997-12-30 US disclosed
EP-0652742-B1 USE OF 3-SUBSTITUTED PARA-AMINOPHENOLS FOR DYEING KERATINOUS FIBRES AND NOVEL SUBSTITUTED 3-PARA-AMINOPHENOLS OREAL (FR) 1997-08-27 EP disclosed
CN-1110048-A Novel 3-substituted para-aminophenols and their use for dyeing keratin fibers OREAL (FR) 1995-10-11 CN disclosed
WO-1994027564-A1 USE OF 3-SUBSTITUTED PARA-AMINOPHENOLS FOR DYEING KERATINOUS FIBRES AND NOVEL SUBSTITUTED 3-PARA-AMINOPHENOLS L'OREAL (FR) 1994-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030181742-A1 Process for the preparation of pregnane derivatives CYP21A2, CYP11B2, CYP17A1 ALDH1A1 1934/4885TSHR 1634/4885TDP1 4556/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.