SCHEMBL8745930

SCHEMBL8745930

CCc1ncncc1C(=O)c1ccccc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.43
CYP3A4 P08684 2/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CTNNB1 P35222 2/20 0.41
WNT3A P56704 2/20 0.41
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329113 0.75 RBP4 (0.44) CNR2CYP3A4HSD17B10KDM4ETSHR
SCHEMBL746794 0.74 LMNA (0.64) CNR2CTNNB1WNT3ALMNAGAA
SCHEMBL28815055 0.73 LMNA (0.62) CNR2CTNNB1WNT3ALMNAGAA
SCHEMBL8828275 0.71 CYP3A4 (0.39) CNR2CYP3A4HSD17B10KDM4ETSHR
SCHEMBL13728541 0.71 CNR2 (0.54) CNR2CTNNB1WNT3ALMNAGAA
SCHEMBL8328355 0.70 GABRP (0.43) KDM4EALDH1A1SMN1; SMN2
SCHEMBL15782804 0.70 SMN1; SMN2 (0.36) CYP3A4KDM4ETSHRTDP1ALDH1A1
SCHEMBL6859050 0.69 HSP90AB1 (0.34) HSD17B10KDM4ETSHRTDP1MAPT
SCHEMBL5990096 0.68 LMNA (0.42) CNR2CTNNB1WNT3ALMNAGAA
SCHEMBL6646161 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5672567-A PRE- AND POST-EMERGENCE ZENECA LIMITED (GB) 1997-09-30 US disclosed
US-5670453-A PYRAZINEARYL COMPOUND ZENECA LIMITED (GB) 1997-09-23 US disclosed
EP-0758323-A1 HERBICIDAL HYDROXYBENZYL-SUBSTITUTED HETEROARYL COMPOUNDS AND DERIVATIVES THEREOF ZENECA LIMITED (GB) 1997-02-19 EP disclosed
WO-1995029898-A1 HERBICIDAL HYDROXYBENZYL-SUBSTITUTED HETEROARYL COMPOUNDS AND DERIVATIVES THEREOF ZENECA LIMITED (GB) 1995-11-09 WO disclosed