SCHEMBL8746248

SCHEMBL8746248

N#Cc1ccc(C(c2ccc(C#N)cc2)c2cnco2)cc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 14/20 0.56
NOTUM Q6P988 1/20 0.40
CYP11B2 P19099 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP11B1 P15538 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
KEAP1 Q14145 1/20 0.35
NAMPT P43490 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CYP2A6 P11509 1/20 0.33
CA12 O43570 1/20 0.33
CA2 P00918 1/20 0.33
CA3 P07451 1/20 0.33
CA6 P23280 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4078028 0.73 CYP19A1 (0.68) CYP19A1CYP11B2CYP3A4CYP11B1TSHR
SCHEMBL2355389 0.72 CYP19A1 (1.00) CYP19A1CYP11B2CYP3A4CYP11B1TSHR
SCHEMBL8700864 0.71 CYP19A1 (0.69) CYP19A1CYP11B2CYP3A4CYP11B1TSHR
SCHEMBL2921542 0.70 KEAP1 (0.68) NOTUMCYP11B2CYP3A4CYP11B1KEAP1
SCHEMBL8746229 0.68 CYP19A1 (0.56) CYP19A1NOTUMCYP11B2CYP3A4CYP11B1
SCHEMBL9790964 0.68 CYP19A1 (1.00) CYP19A1CYP11B2CYP3A4CYP11B1ALDH1A1
SCHEMBL2354875 0.68 CYP19A1 (1.00) CYP19A1CYP11B2CYP3A4CYP11B1ALDH1A1
SCHEMBL2356831 0.67 CYP19A1 (0.54) CYP19A1CYP11B2CYP3A4CYP11B1TSHR
Hydrochloric Acid SCHEMBL1507785 0.67 CYP19A1 (0.97) CYP19A1CYP11B2CYP3A4CYP11B1ALDH1A1
SCHEMBL1343704 0.66 CYP19A1 (0.63) CYP19A1TSHRALDH1A1CYP2A6CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0477141-B1 Heteroarylmethylbenzols aromatase inhibitors CIBA GEIGY AG (CH) 1997-02-26 EP disclosed
US-5378721-A AROMATASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1995-01-03 US disclosed
US-5246952-A Antitumor agents CIBA-GEIGY CORPORATION (US) 1993-09-21 US disclosed
EP-0477141-A1 Heteroarylmethylbenzols aromatase inhibitors CIBA-GEIGY AG (CH) 1992-03-25 EP disclosed