SCHEMBL8746252

SCHEMBL8746252

N#Cc1ccc(C(O)c2cncs2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 10/20 0.44
FNTA P49354 3/20 0.42
FNTB P49356 3/20 0.42
MYC P01106 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP11B1 P15538 1/20 0.36
TSHR P16473 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP2C19 P33261 1/20 0.36
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35
BRD4 O60885 1/20 0.34
CA12 O43570 1/20 0.34
CA2 P00918 1/20 0.34
CA3 P07451 1/20 0.34
CA6 P23280 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
GSK3B P49841 1/20 0.34
PGR P06401 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2356831 0.83 CYP19A1 (0.54) CYP19A1FNTAFNTBMYCCYP3A4
SCHEMBL31040275 0.78 TSHR (0.36) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL14033955 0.78 SLC6A3 (0.45) CYP19A1TSHR
SCHEMBL28752724 0.78 SLC6A3 (0.41) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL2974022 0.78 SLC6A3 (0.45) CYP19A1CYP11B1TSHRCYP11B2
SCHEMBL8633394 0.78 SMN1; SMN2 (0.48) TSHR
SCHEMBL691258 0.74 CA2 (0.52) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL30251242 0.72 CYP19A1 (0.53) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL17338939 0.72 CYP19A1 (0.53) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL8634094 0.71 SLC6A2 (0.40) CYP3A4BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0477141-B1 Heteroarylmethylbenzols aromatase inhibitors CIBA GEIGY AG (CH) 1997-02-26 EP disclosed
US-5378721-A AROMATASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1995-01-03 US disclosed
US-5246952-A Antitumor agents CIBA-GEIGY CORPORATION (US) 1993-09-21 US disclosed
EP-0477141-A1 Heteroarylmethylbenzols aromatase inhibitors CIBA-GEIGY AG (CH) 1992-03-25 EP disclosed