SCHEMBL8747158

SCHEMBL8747158

COc1cc2c(cc1OCc1ccccc1)C(C1(c3ccccc3SC)CCC1)NC=C2

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
CISD1 Q9NZ45 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
CHRNA7 P36544 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747329 0.81 PKM (0.45) MEN1KMT2AADRA1DADRA1AADRA1B
SCHEMBL8747178 0.76 CHRNA7 (0.48) ADRA1DADRA1AADRA1BCHRNA7
SCHEMBL17375771 0.72 NPC1 (0.42) MEN1KMT2ASIRT2SMN1; SMN2CHRNA7
SCHEMBL8747147 0.69 PKM (0.46) MEN1KMT2ACHRNA7
SCHEMBL8747269 0.66 KDM4E (0.45) MEN1KMT2ACHRNA7
SCHEMBL8747338 0.65 PKM (0.44) MEN1KMT2ACHRNA7
SCHEMBL8746992 0.64 MEN1 (0.46) MEN1KMT2ACHRNA7
Bromide SCHEMBL8747077 0.64 MEN1 (0.45) MEN1KMT2ACHRNA7
SCHEMBL8747218 0.63 CHRNA7 (0.50) CHRNA7
SCHEMBL29993463 0.62 CHRNA7 (0.45) SMN1; SMN2CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed