SCHEMBL8747251

SCHEMBL8747251

CN1CCc2cc([N+](=O)[O-])c(O)cc2C1C1(c2ccccc2)CCC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.40
DRD1 P21728 4/20 0.39
DRD2 P14416 3/20 0.39
HIF1A Q16665 2/20 0.38
STS P08842 2/20 0.37
MAOA P21397 1/20 0.36
CYP19A1 P11511 1/20 0.36
MAPK1 P28482 1/20 0.36
THPO P40225 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MTOR P42345 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL8747274 0.97 SIRT6 (0.38) SIRT6DRD1DRD2HIF1ASTS
SCHEMBL8747006 0.85 MAOA (0.50) DRD1DRD2HIF1AMAOAMAPK1
SCHEMBL8747278 0.85 POLB (0.39) SIRT6
Bromide SCHEMBL8747268 0.84 KDM4E (0.49) DRD1DRD2HIF1AMAOAMAPK1
SCHEMBL8747355 0.83 MAOA (0.50) DRD1DRD2HIF1AMAOAMAPK1
SCHEMBL8747054 0.82 MAOA (0.49) DRD1DRD2HIF1AMAOAMAPK1
SCHEMBL8747056 0.81 DRD1 (0.60) DRD1DRD2MAPK1THPOHSD17B10
SCHEMBL8747233 0.81 DRD1 (0.52) DRD1DRD2MAPK1HSD17B10
SCHEMBL8747186 0.81 DRD1 (0.43) DRD1DRD2HIF1AMAOAMAPK1
SCHEMBL8747280 0.81 MAOA (0.52) DRD1DRD2HIF1AMAOAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed