SCHEMBL8747282

SCHEMBL8747282

COc1cc2c(cc1Cl)CCNC2C1(c2ccccc2)CCC1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.51
PKM P14618 1/20 0.49
HTR2A P28223 4/20 0.47
HTR2C P28335 4/20 0.47
HTR2B P41595 4/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP3A4 P08684 1/20 0.41
MAOA P21397 2/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747312 0.84 SLC6A9 (0.65) SLC6A9PKMMEN1KMT2ACYP3A4
Hydrochloric Acid SCHEMBL8747055 0.83 PKM (0.54) SLC6A9PKMMEN1KMT2AMAOA
SCHEMBL9298751 0.81 SLC6A9 (0.54) SLC6A9PKMHTR2AHTR2CHTR2B
SCHEMBL989918 0.81 SLC6A9 (0.60) SLC6A9PKMHTR2AHTR2CHTR2B
SCHEMBL8747203 0.80 PKM (0.47) SLC6A9PKMHTR2AHTR2CHTR2B
SCHEMBL8747118 0.79 PKM (0.54) SLC6A9PKMMEN1KMT2ACYP3A4
SCHEMBL8747215 0.77 PKM (0.54) SLC6A9PKMHTR2AHTR2CHTR2B
SCHEMBL8747147 0.76 PKM (0.46) SLC6A9PKMHTR2AHTR2CMEN1
SCHEMBL989030 0.76 SLC6A9 (0.54) SLC6A9PKMCYP3A4MAOA
SCHEMBL8747148 0.76 PKM (0.55) SLC6A9PKMHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed