SCHEMBL8747148

SCHEMBL8747148

COc1cc2c(cc1OC)C(C1(c3ccccc3Br)CCC1)NCC2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.55
KMT2A Q03164 5/20 0.50
MEN1 O00255 3/20 0.50
MAOA P21397 2/20 0.46
TSHR P16473 1/20 0.46
DRD1 P21728 1/20 0.42
DRD5 P21918 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
SLC6A9 P48067 1/20 0.41
GAA P10253 1/20 0.41
BCHE P06276 1/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747254 0.87 PKM (0.46) PKMKMT2AMEN1MAOATSHR
SCHEMBL8747258 0.86 PKM (0.44) PKMKMT2AMEN1MAOATSHR
SCHEMBL27349849 0.85 PKM (0.43) PKMKMT2AMEN1DRD1DRD5
SCHEMBL8747203 0.80 PKM (0.47) PKMKMT2AMEN1MAOATSHR
SCHEMBL8747215 0.79 PKM (0.54) PKMKMT2AMEN1MAOATSHR
SCHEMBL8747118 0.79 PKM (0.54) PKMKMT2AMEN1MAOATSHR
Hydrochloric Acid SCHEMBL8747055 0.79 PKM (0.54) PKMKMT2AMEN1MAOATSHR
SCHEMBL8747147 0.78 PKM (0.46) PKMKMT2AMEN1SLC6A9HTR2A
SCHEMBL8747173 0.78 MAOA (0.47) KMT2AMEN1MAOADRD1DRD5
SCHEMBL8747312 0.77 SLC6A9 (0.65) PKMKMT2AMEN1MAOATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed