Oxalic Acid

Oxalic Acid

SCHEMBL8747351

COc1cc2c(cc1O)C(C1(c3ccc(Cl)cc3)CCC1)N(C)CC2.O=C(O)C(=O)O

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 5/20 0.52
DRD2 P14416 3/20 0.52
TP53 P04637 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
DRD5 P21918 2/20 0.46
MAOA P21397 2/20 0.43
TRPV1 Q8NER1 1/20 0.42
GRIN2D O15399 4/20 0.42
GRIN3B O60391 4/20 0.42
GRIN1 Q05586 4/20 0.42
GRIN2A Q12879 4/20 0.42
GRIN2B Q13224 4/20 0.42
GRIN2C Q14957 4/20 0.42
GRIN3A Q8TCU5 4/20 0.42
KCNH2 Q12809 1/20 0.42
NR1I2 O75469 1/20 0.42
PTGS2 P35354 1/20 0.42
OPRK1 P41145 1/20 0.42
SLC6A3 Q01959 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747191 0.95 DRD1 (0.56) DRD1DRD2TP53TSHRMAPK1
SCHEMBL8747012 0.88 DRD1 (0.50) DRD1DRD2TP53TSHRMAPK1
Oxalic Acid SCHEMBL8747231 0.87 DRD2 (0.56) DRD1DRD2MAOAKCNH2
SCHEMBL8747029 0.86 DRD1 (0.50) DRD1DRD2TP53TSHRMAPK1
SCHEMBL8747354 0.86 TRPV1 (0.48) DRD1DRD2TP53TSHRMAPK1
SCHEMBL8747074 0.85 DRD1 (0.49) DRD1DRD2TP53TSHRMAPK1
SCHEMBL8747405 0.85 MAOA (0.47) DRD1DRD2TP53TSHRMAPK1
Bromide SCHEMBL8747099 0.84 MAOA (0.46) DRD1DRD2TP53TSHRMAPK1
SCHEMBL8747142 0.83 DRD1 (0.53) DRD1DRD2TSHRMAPK1DRD5
SCHEMBL8747336 0.83 TP53 (0.51) DRD1DRD2TP53TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed