SCHEMBL874737

SCHEMBL874737

CCn1c(N)nc2nc[nH]c2c1=O

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 12/20 0.56
ADORA2B P29275 8/20 0.56
PDE4A P27815 12/20 0.54
PDE4B Q07343 12/20 0.54
PDE4C Q08493 12/20 0.54
PDE4D Q08499 12/20 0.54
PNP P00491 1/20 0.45
DPP4 P27487 1/20 0.42
ADORA3 P0DMS8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL667797 0.88 PDE4A (0.60) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL6272735 0.85 PDE4A (0.59) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL1047660 0.84 PNP (0.45) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL28071828 0.84 PNP (0.45) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL1767750 0.84 ADORA2A (0.47) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL8522275 0.84 ADORA2B (0.61) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL5504400 0.84 ADORA2A (0.59) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL2343362 0.84 ADORA2A (0.44) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL8536009 0.83 ADORA2B (0.64) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL6272301 0.83 ADORA2B (0.64) ADORA2AADORA2BPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 112 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9725474-B2 Modified nucleic acid TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-08 US claimed
EP-1419247-A2 METHOD FOR THE PRODUCTION OF NUCLEIC ACIDS CONSISTING OF STOCHASTICALLY COMBINED PARTS OF SOURCE NUCLEIC ACIDS Direvo Biotech AG (DE) 2004-05-19 EP claimed
WO-2003012100-A2 METHOD FOR THE PRODUCTION OF NUCLEIC ACIDS CONSISTING OF STOCHASTICALLY COMBINED PARTS OF SOURCE NUCLEIC ACIDS DIREVO BIOTECH AG (DE) 2003-02-13 WO claimed
EP-4658084-A1 FOOD COMPOSITION Unilever IP Holdings B.V. (NL) 2025-12-10 EP disclosed
EP-4658754-A1 ALGAE BIOMASS Algenuity BV (NL) 2025-12-10 EP disclosed
EP-4658753-A1 CHLORELLA MICROALGAE Algenuity BV (NL) 2025-12-10 EP disclosed
EP-4658093-A1 FOOD COMPOSITION COMPRISING CHLOROPHYLL-DEFICIENT CHLORELLA BIOMASS WITH HIGH PROTEIN CONTENT >50WT% Unilever IP Holdings B.V. (NL) 2025-12-10 EP disclosed
WO-2025082420-A1 AQUEOUS EMULSION, METHOD FOR PREPARING THE SAME, COATING COMPOSITION AND ARTICLE GUANGDONG HUARUN PAINTS CO., LTD. (CN) 2025-04-24 WO disclosed
EP-4522753-A2 DOUBLE STRANDED DNA COMPOSITIONS AND RELATED METHODS Flagship Pioneering Innovations VII, LLC (US) 2025-03-19 EP disclosed
US-20250027033-A1 MODIFIED STRAINS OF CHLORELLA VULGARIS AND METHOD OF PRODUCTION ALGENUITY HOLDINGS LTD (GB) 2025-01-23 US disclosed
WO-2024178065-A2 CRIPPLED CORONAVIRUS: 5'-POLYU TARGETED OLIGO PREVENTS DEVELOPMENT OF INFECTIOUS VIRIONS HOWARD UNIVERSITY (US) 2024-08-29 WO disclosed
US-6303618-B1 ADMINISTERING PURINE COMPOUND WHICH INHIBITS CYCLIC DEPENDENT KINASE ACTIVITY FOR THERAPY OF TUMOR OR OTHER CELL PROLIFERATION DISORDER CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2001-10-16 US disclosed
WO-2000017220-A1 ANTISENSE MODULATION OF FAN EXPRESSION ISIS PHARMACEUTICALS, INC. (US) 2000-03-30 WO disclosed
WO-1999002162-A9 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RES CAMPAIGN TECH (GB) 1999-07-29 WO disclosed
EP-0846772-A1 Multifunctional ligand system for cell-specific transfer of nucleic acid HOECHST AKTIENGESELLSCHAFT (DE) 1998-06-10 EP disclosed
EP-0666903-A4 INSULIN-DEPENDENT YEAST OR FUNGI. MCKENZIE MAUREEN A (US) 1997-06-04 EP disclosed
EP-0702683-A1 06-SUBSTITUTED GUANINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN TREATING TUMOUR CELLS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1996-03-27 EP disclosed
EP-0666903-A1 INSULIN-DEPENDENT YEAST OR FUNGI McKENZIE, Maureen A. (US) 1995-08-16 EP disclosed
WO-1994007994-A9 INSULIN-DEPENDENT YEAST OR FUNGI 1994-06-09 WO disclosed
WO-1994007994-A1 INSULIN-DEPENDENT YEAST OR FUNGI MCKENZIE MAUREEN A (US) 1994-04-14 WO disclosed