SCHEMBL875016

SCHEMBL875016

CCCn1nc(-c2ccc(NC(=O)NCc3ccc(N)nc3)cc2)cc1C(=O)NCCN1CCS(=O)(=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 7/20 0.41
HDAC1 Q13547 1/20 0.41
KIT P10721 1/20 0.40
JAK2 O60674 2/20 0.38
CPB1 P15086 1/20 0.36
ROCK2 O75116 1/20 0.36
ATR Q13535 2/20 0.36
ACVR1 Q04771 1/20 0.35
AURKA O14965 1/20 0.35
AURKB Q96GD4 1/20 0.35
KDR P35968 1/20 0.35
FLT3 P36888 1/20 0.35
CNR1 P21554 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874907 0.93 NAMPT (0.47) NAMPTHDAC1KITJAK2ATR
SCHEMBL875705 0.85 NAMPT (0.47) NAMPTHDAC1CPB1ROCK2
SCHEMBL875445 0.84 NAMPT (0.46) NAMPTHDAC1KITJAK2ATR
SCHEMBL875943 0.82 NAMPT (0.48) NAMPTHDAC1KITJAK2ATR
SCHEMBL874894 0.82 NAMPT (0.46) NAMPTHDAC1KITJAK2ATR
SCHEMBL3051319 0.81 NAMPT (0.40) NAMPTHDAC1KITJAK2ROCK2
SCHEMBL874909 0.80 CHRNA7 (0.47) NAMPTHDAC1KITJAK2ATR
SCHEMBL875170 0.80 HDAC1 (0.41) NAMPTHDAC1KITJAK2ROCK2
SCHEMBL875967 0.78 NAMPT (0.40) NAMPTHDAC1KITCPB1ROCK2
SCHEMBL874781 0.76 HDAC6 (0.48) NAMPTHDAC1CPB1ROCK2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed