SCHEMBL875170

SCHEMBL875170

CCNc1cc(-c2ccc(NC(=O)NCc3ccc(N)nc3)cc2)sc1C(=O)NCCN1CCS(=O)(=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.41
NAMPT P43490 7/20 0.40
KIT P10721 1/20 0.39
ROCK2 O75116 2/20 0.38
LIMK1 P53667 1/20 0.38
MAP3K7 O43318 1/20 0.36
RXFP1 Q9HBX9 1/20 0.34
CNR1 P21554 1/20 0.34
IKBKB O14920 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL875381 0.92 NAMPT (0.47) HDAC1NAMPTKITJAK2JAK1
SCHEMBL875967 0.87 NAMPT (0.40) HDAC1NAMPTKITROCK2LIMK1
SCHEMBL10070169 0.86 NAMPT (0.36) HDAC1NAMPTLIMK1MAP3K7RXFP1
SCHEMBL874891 0.83 HDAC1 (0.50) HDAC1NAMPTROCK2IKBKB
SCHEMBL875667 0.82 CD274 (0.42) MAP3K7JAK2JAK1TYK2JAK3
SCHEMBL3051319 0.81 NAMPT (0.40) HDAC1NAMPTKITROCK2JAK2
SCHEMBL875067 0.81 NAMPT (0.44) HDAC1NAMPT
SCHEMBL875016 0.80 NAMPT (0.41) HDAC1NAMPTKITROCK2CNR1
SCHEMBL874755 0.79 NAMPT (0.47) HDAC1NAMPTKIT
SCHEMBL486122 0.75 PIK3CA (0.39) HDAC1KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed