SCHEMBL875067

SCHEMBL875067

Nc1ccc(CNC(=O)Nc2ccc(-c3nc(Nc4ccccc4)c(C(=O)NCCN4CCS(=O)(=O)CC4)s3)cc2)cn1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 10/20 0.44
HDAC1 Q13547 1/20 0.43
ATR Q13535 3/20 0.39
BTK Q06187 1/20 0.38
WNT3A P56704 1/20 0.37
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
AURKA O14965 1/20 0.37
AURKB Q96GD4 1/20 0.37
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874813 0.92 NAMPT (0.48) NAMPTHDAC1ATRMEN1POLB
SCHEMBL875967 0.89 NAMPT (0.40) NAMPTHDAC1ATR
SCHEMBL874755 0.81 NAMPT (0.47) NAMPTHDAC1ATRMEN1POLB
SCHEMBL875170 0.81 HDAC1 (0.41) NAMPTHDAC1
SCHEMBL874266 0.79 NAMPT (0.49) NAMPTHDAC1ATRMEN1POLB
SCHEMBL3051507 0.78 ATR (0.50) NAMPTHDAC1ATRMEN1POLB
SCHEMBL3051319 0.77 NAMPT (0.40) NAMPTHDAC1ATR
SCHEMBL874795 0.76 NAMPT (0.47) NAMPTHDAC1ATR
SCHEMBL883091 0.76 NAMPT (0.36) NAMPTHDAC1
SCHEMBL875016 0.75 NAMPT (0.41) NAMPTHDAC1ATRAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed