SCHEMBL8750729

SCHEMBL8750729

N#Cc1cncc(NCc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.48
CYP2C19 P33261 3/20 0.48
TSHR P16473 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CHRNB2 P17787 1/20 0.47
CHRNA4 P43681 1/20 0.47
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47
ABCB1 P08183 3/20 0.46
ABCG2 Q9UNQ0 3/20 0.46
VNN1 O95497 2/20 0.46
EGLN2 Q96KS0 1/20 0.45
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
LTA4H P09960 1/20 0.45
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2038512 0.80 RAB9A (0.52) TSHRCYP2D6KDM4EHPGDALDH1A1
SCHEMBL1680823 0.79 LMNA (0.57) CYP1A2CYP2C19TSHRCYP3A4CYP2D6
SCHEMBL510619 0.76 HTT (0.58) CYP1A2TSHRCYP2D6ABCB1ABCG2
SCHEMBL22191457 0.76 KDM4E (0.50) CYP1A2CYP2C19CYP3A4CYP2D6ABCB1
SCHEMBL22191849 0.76 LRRK2 (0.49) CYP1A2CYP2C19TSHRCYP3A4CYP2D6
SCHEMBL2064845 0.76 SMN1; SMN2 (0.54) CHRNB2CHRNA4GABRG2GABRB3GABRA5
SCHEMBL21591750 0.76 LTA4H (0.49) CHRNB2CHRNA4KDM4EHPGDLTA4H
SCHEMBL6772345 0.76 KCNH2 (0.56) CHRNB2CHRNA4HPGDLTA4HKCNH2
SCHEMBL13743125 0.76 KCNH2 (0.56) CYP1A2CYP2C19CYP3A4CYP2D6HSD17B10
SCHEMBL8750751 0.75 CHEK1 (0.42) GABRG2GABRB3GABRA5GABRA3EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1043760-C \"Pyridinecarboximidamide compounds and the use thereof\ KIRN BEER KABUSHIKI KAISHA (JP) 1999-06-23 CN disclosed
EP-0634400-B1 PYRIDINECARBOXIMIDAMIDE COMPOUND AND USE THEREOF KIRIN BREWERY (JP) 1997-04-02 EP disclosed
US-5508293-A TREATING HYPERTENSION, ANGINA PECTORIS KIRIN BEER KABUSHIKI KAISHA (JP) 1996-04-16 US disclosed
EP-0634400-A1 PYRIDINECARBOXIMIDAMIDE COMPOUND AND USE THEREOF KIRIN BEER KABUSHIKI KAISHA (JP) 1995-01-18 EP disclosed
CN-1077949-A Pyridine carboxy imido acid amide compound and application thereof KIRIN BREWERY (JP) 1993-11-03 CN disclosed