SCHEMBL875402

SCHEMBL875402

CC(C)n1nc(-c2ccc(NC(=O)NCc3ccc(N)nc3)cc2)cc1C(=O)NC1CC1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 7/20 0.45
HDAC1 Q13547 3/20 0.45
HDAC6 Q9UBN7 1/20 0.40
KLKB1 P03952 1/20 0.40
ACVR1 Q04771 1/20 0.38
ROCK2 O75116 2/20 0.38
CPB1 P15086 1/20 0.37
PPIB P23284 1/20 0.37
DGAT1 O75907 1/20 0.37
BRD4 O60885 1/20 0.36
KIT P10721 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL875709 0.97 NAMPT (0.44) NAMPTHDAC1HDAC6KLKB1ACVR1
SCHEMBL874781 0.87 HDAC6 (0.48) NAMPTHDAC1HDAC6ROCK2CPB1
SCHEMBL875615 0.87 NAMPT (0.45) NAMPTHDAC1HDAC6ROCK2CPB1
SCHEMBL875268 0.82 NAMPT (0.40) NAMPTHDAC6ACVR1BRD4KIT
SCHEMBL875269 0.82 NAMPT (0.40) NAMPTHDAC6ACVR1BRD4KIT
SCHEMBL874150 0.77 HDAC6 (0.48) HDAC6ACVR1BRD4
SCHEMBL875445 0.76 NAMPT (0.46) NAMPTHDAC1KIT
SCHEMBL3050217 0.76 HDAC1 (0.47) NAMPTHDAC1ROCK2
SCHEMBL882752 0.75 NAMPT (0.46) NAMPTHDAC1KLKB1CPB1PPIB
SCHEMBL875705 0.75 NAMPT (0.47) NAMPTHDAC1ROCK2CPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed