SCHEMBL875709

SCHEMBL875709

CC(C)n1nc(-c2ccc(NC(=O)NCc3ccc(N)nc3)cc2)cc1C(=O)NC1CCCC1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 7/20 0.44
HDAC1 Q13547 1/20 0.43
KIT P10721 1/20 0.41
HDAC6 Q9UBN7 1/20 0.39
ACVR1 Q04771 1/20 0.38
CARM1 Q86X55 1/20 0.38
PPIB P23284 1/20 0.38
KLKB1 P03952 1/20 0.37
FAAH O00519 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
EPHX1 P07099 1/20 0.37
ROCK2 O75116 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL875402 0.97 NAMPT (0.45) NAMPTHDAC1KITHDAC6ACVR1
SCHEMBL875615 0.85 NAMPT (0.45) NAMPTHDAC1HDAC6ROCK2
SCHEMBL874781 0.85 HDAC6 (0.48) NAMPTHDAC1HDAC6ROCK2
SCHEMBL875268 0.79 NAMPT (0.40) NAMPTKITHDAC6ACVR1NPC1
SCHEMBL875269 0.79 NAMPT (0.40) NAMPTKITHDAC6ACVR1NPC1
SCHEMBL875445 0.76 NAMPT (0.46) NAMPTHDAC1KIT
SCHEMBL3042675 0.76 NAMPT (0.45) NAMPTHDAC1KITACVR1EPHX1
SCHEMBL874150 0.74 HDAC6 (0.48) HDAC6ACVR1
SCHEMBL875705 0.73 NAMPT (0.47) NAMPTHDAC1ROCK2
SCHEMBL874894 0.73 NAMPT (0.46) NAMPTHDAC1KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed