SCHEMBL875487

SCHEMBL875487

CCNc1nc(-c2ccc(NC(=O)NCc3ccc(N)nc3)cc2)sc1C(=O)NCCOC

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.45
NAMPT P43490 11/20 0.44
ROCK2 O75116 4/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPKAPK2 P49137 1/20 0.37
PPARA Q07869 1/20 0.37
MTOR P42345 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL875947 0.88 PPARA (0.49) HDAC1NAMPTALDH1A1POLBSMN1; SMN2
SCHEMBL874763 0.88 NAMPT (0.43) HDAC1NAMPTROCK2ALDH1A1POLB
SCHEMBL874755 0.86 NAMPT (0.47) HDAC1NAMPTPOLB
SCHEMBL875702 0.85 NAMPT (0.44) HDAC1NAMPTROCK2ALDH1A1POLB
SCHEMBL875967 0.84 NAMPT (0.40) HDAC1NAMPTROCK2PPARA
SCHEMBL3057949 0.84 HDAC1 (0.45) HDAC1NAMPTROCK2MAPKAPK2MTOR
SCHEMBL874752 0.77 NAMPT (0.52) HDAC1NAMPTALDH1A1POLBSMN1; SMN2
SCHEMBL3054524 0.75 HDAC1 (0.46) HDAC1NAMPTROCK2POLB
SCHEMBL882700 0.75 POLB (0.60) NAMPTALDH1A1POLB
SCHEMBL874813 0.74 NAMPT (0.48) HDAC1NAMPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed