SCHEMBL875758

SCHEMBL875758

CN(C(=O)c1ccc2c(c1)CCC2N1C=NC=C(OC(=O)O)C1)C1CCN(c2ccncc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F10 P00742 4/20 0.34
CCR5 P51681 1/20 0.34
GHSR Q92847 5/20 0.33
MCHR1 Q99705 1/20 0.33
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
ABL1 P00519 2/20 0.32
PDGFRB P09619 2/20 0.32
KIT P10721 2/20 0.32
ROCK2 O75116 1/20 0.32
POLB P06746 1/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878508 0.94 F10 (0.34) F10CCR5MCHR1JAK2JAK1
SCHEMBL876131 0.89 POLB (0.34) F10CCR5MCHR1JAK2JAK1
SCHEMBL876268 0.86 F10 (0.34) F10CCR5MCHR1ROCK2POLB
SCHEMBL878362 0.84 TLR9 (0.36) F10JAK2JAK1POLB
SCHEMBL875680 0.79 F10 (0.33) F10CCR5GHSRMCHR1JAK2
SCHEMBL875757 0.77 CCR5 (0.35) F10CCR5GHSRMCHR1JAK2
SCHEMBL875679 0.76 F10 (0.34) F10CCR5GHSRMCHR1JAK2
SCHEMBL786045 0.76 CCR5 (0.42) F10CCR5MCHR1JAK2JAK1
SCHEMBL876715 0.76 CCR5 (0.37) F10CCR5MCHR1JAK2JAK1
SCHEMBL878284 0.75 F10 (0.39) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed