SCHEMBL876268

SCHEMBL876268

CN(C(=O)c1ccc2c(c1)C(N1C=NC=C(OC(=O)O)C1)CCO2)C1CCN(c2ccncc2)CC1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F10 P00742 5/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CCR5 P51681 1/20 0.33
KDM4C Q9H3R0 2/20 0.31
KDM6B O15054 1/20 0.31
CHRM1 P11229 1/20 0.30
MCHR1 Q99705 1/20 0.30
ROCK2 O75116 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878508 0.87 F10 (0.34) F10CCR5MCHR1POLB
SCHEMBL876131 0.86 POLB (0.34) F10CCR5MCHR1POLB
SCHEMBL875758 0.86 F10 (0.34) F10CCR5MCHR1ROCK2POLB
SCHEMBL876160 0.80 F10 (0.33) F10NPC1RAB9ACCR5MCHR1
SCHEMBL876267 0.78 F10 (0.36) F10NPC1RAB9ACCR5KDM4C
SCHEMBL878362 0.78 TLR9 (0.36) F10POLB
SCHEMBL876159 0.77 NPC1 (0.35) F10NPC1RAB9ACCR5KDM4C
SCHEMBL784870 0.77 F10 (0.42) F10NPC1RAB9ACCR5ROCK2
SCHEMBL784756 0.74 F10 (0.40) F10NPC1RAB9ACCR5KDM4C
SCHEMBL785183 0.73 F10 (0.39) F10NPC1RAB9ACCR5ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed