SCHEMBL878362

SCHEMBL878362

Cc1cc(N2CCC(N(C)C(=O)c3ccc4c(c3)C(N3C=NC=C(OC(=O)O)C3)CC4)CC2)cc(C)n1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
F10 P00742 1/20 0.34
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
JAK2 O60674 6/20 0.31
JAK1 P23458 6/20 0.31
POLB P06746 1/20 0.31
DRD2 P14416 1/20 0.31
MRGPRX2 Q96LB1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878508 0.90 F10 (0.34) F10ADORA2AADORA1JAK2JAK1
SCHEMBL876131 0.86 POLB (0.34) F10JAK2JAK1POLB
SCHEMBL875758 0.84 F10 (0.34) F10JAK2JAK1POLB
SCHEMBL878405 0.82 TLR9 (0.37) TLR9TLR8TLR7F10ADORA2A
SCHEMBL878327 0.79 TLR9 (0.36) TLR9TLR8TLR7F10ADORA2A
SCHEMBL876268 0.78 F10 (0.34) F10POLB
SCHEMBL878326 0.77 TLR9 (0.39) TLR9TLR8TLR7F10ADORA2A
SCHEMBL785591 0.77 F10 (0.44) TLR9TLR8TLR7F10ADORA2A
SCHEMBL784885 0.75 TLR9 (0.42) TLR9TLR8TLR7F10ADORA2A
SCHEMBL784539 0.75 TLR9 (0.43) TLR9TLR8TLR7F10ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed