SCHEMBL8759101

SCHEMBL8759101

CS(=O)(=O)c1ccccc1-n1cccn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 3/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 1/20 0.42
G6PD P11413 1/20 0.42
DRD2 P14416 1/20 0.41
CREBBP Q92793 1/20 0.41
KAT6A Q92794 1/20 0.40
ACLY P53396 1/20 0.39
CHRM1 P11229 1/20 0.39
ADRA2A P08913 1/20 0.38
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29484301 0.83 MAPK1 (0.49) MAPK1NPC1ALDH1A1LMNAMEN1
SCHEMBL15266274 0.83 MAPK1 (0.49) MAPK1NPC1ALDH1A1LMNAMEN1
SCHEMBL621024 0.83 MAPK1 (0.49) MAPK1NPC1ALDH1A1LMNAMEN1
SCHEMBL10547713 0.83 MAPK1 (0.49) MAPK1NPC1ALDH1A1LMNAMEN1
SCHEMBL28293040 0.80 KMT2A (0.40) MAPK1NPC1ALDH1A1LMNAHTT
SCHEMBL28294729 0.80 MAPT (0.37) MAPK1NPC1ALDH1A1LMNATP53
SCHEMBL4341886 0.77 MAPK1 (0.67) MAPK1NPC1ALDH1A1LMNAHTT
SCHEMBL28425880 0.76 MAPT (0.41) MAPK1NPC1ALDH1A1LMNAMEN1
SCHEMBL30183430 0.76 MAPK1 (0.49) MAPK1NPC1ALDH1A1LMNAMEN1
SCHEMBL8662730 0.75 NPC1 (0.42) MAPK1NPC1ALDH1A1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108477173-A Heterocyclic compound as insecticide 拜耳农作物科学股份公司 2018-09-04 CN disclosed
CN-105101800-B Heterocyclic Compounds as Pesticides 拜耳农作物科学股份公司 2018-04-13 CN disclosed
CN-102171213-A Pyrazolo [3, 4] pyrimidin-4-yl derivatives and their uses to treat diabetes and obesity ASTRAZENECA AB 2011-08-31 CN disclosed
EP-0772597-A1 3,4-SUBSTITUTED PYRAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-05-14 EP disclosed
WO-1996003385-A1 3,4-SUBSTITUTED PYRAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed