SCHEMBL28294729

SCHEMBL28294729

CS(=O)(=O)c1c[c]ccc1-n1cccn1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.37
KMT2A Q03164 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
G6PD P11413 1/20 0.37
MAPK1 P28482 2/20 0.36
NPC1 O15118 1/20 0.36
ACLY P53396 1/20 0.34
KAT6A Q92794 1/20 0.33
TDO2 P48775 1/20 0.33
NOTUM Q6P988 1/20 0.33
CYP46A1 Q9Y6A2 1/20 0.32
POLB P06746 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8759101 0.80 MAPK1 (0.49) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL28293040 0.73 KMT2A (0.40) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL29001798 0.73 ALDH1A1 (0.42) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL161297 0.73 ALDH1A1 (0.42) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL4878068 0.73 NOTUM (0.44) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL7237526 0.71 KDM4E (0.40) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL21988636 0.71 KDM4E (0.40) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL28425880 0.70 MAPT (0.41) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL27945389 0.70 ALDH1A1 (0.42) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL27934781 0.70 TDO2 (0.44) MAPTKMT2AKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109694351-A Benzo-aza * derivative, preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2019-04-30 CN disclosed