SCHEMBL8760280

SCHEMBL8760280

CC(C)N1C(=O)C(NC(=O)Cc2ccc(Cl)c(Cl)c2)N=C(c2ccccc2)c2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OXTR P30559 7/20 0.58
KCNH2 Q12809 2/20 0.56
CCKBR P32239 5/20 0.54
PSEN1 P49768 2/20 0.51
PSEN2 P49810 2/20 0.51
APH1B Q8WW43 2/20 0.51
NCSTN Q92542 2/20 0.51
APH1A Q96BI3 2/20 0.51
PSENEN Q9NZ42 2/20 0.51
GSAP A4D1B5 1/20 0.51
RAMP1 O60894 2/20 0.49
CALCRL Q16602 2/20 0.49
CCKAR P32238 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8761096 1.00 OXTR (0.58) OXTRKCNH2CCKBRPSEN1PSEN2
SCHEMBL8760279 0.89 KCNH2 (0.60) OXTRKCNH2CCKBRPSEN1PSEN2
SCHEMBL8760298 0.89 KCNH2 (0.69) OXTRKCNH2CCKBRPSEN1PSEN2
SCHEMBL8761607 0.89 KCNH2 (0.69) OXTRKCNH2CCKBRPSEN1PSEN2
SCHEMBL8761397 0.89 KCNH2 (0.69) OXTRKCNH2CCKBRPSEN1PSEN2
SCHEMBL8761602 0.89 CCKBR (0.57) KCNH2CCKBRPSEN1PSEN2APH1B
SCHEMBL8760285 0.85 OXTR (0.64) OXTRKCNH2CCKBRCCKAR
SCHEMBL8761280 0.85 KCNH2 (0.71) KCNH2CCKBRRAMP1CALCRLCCKAR
SCHEMBL8760336 0.84 CCKBR (0.61) OXTRCCKBRCCKAR
SCHEMBL8760328 0.84 CCKBR (0.59) KCNH2CCKBRPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776203-A4 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO INC (US) 1997-12-29 EP disclosed
EP-0776203-A1 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO. INC. (US) 1997-06-04 EP disclosed
US-5633251-A N-2,3-dihydro-1-(2-propyl)-2-oxo-5-phenyl-1h-1,4-benzodiazepines MERCK & CO., INC. (US) 1997-05-27 US disclosed
WO-1996005827-A1 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO., INC. (US) 1996-02-29 WO disclosed