SCHEMBL8760285

SCHEMBL8760285

CCCN1C(=O)C(NC(=O)Cc2ccc(Cl)c(Cl)c2)N=C(c2ccccc2)c2ccccc21

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OXTR P30559 8/20 0.64
KCNH2 Q12809 3/20 0.61
CCKBR P32239 8/20 0.56
CCKAR P32238 2/20 0.53
NOTCH1 P46531 1/20 0.51
RBPJ Q06330 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8760307 0.89 KCNH2 (0.76) OXTRKCNH2CCKBRCCKARNOTCH1
SCHEMBL8462710 0.87 KCNH2 (0.81) OXTRKCNH2
SCHEMBL8761096 0.85 OXTR (0.58) OXTRKCNH2CCKBRCCKAR
SCHEMBL8760280 0.85 OXTR (0.58) OXTRKCNH2CCKBRCCKAR
SCHEMBL8761589 0.78 KCNH2 (0.80) OXTRKCNH2CCKBRCCKARNOTCH1
SCHEMBL9866216 0.78 CCKBR (0.76) OXTRKCNH2CCKBRCCKAR
SCHEMBL8846371 0.77 KCNH2 (0.79) OXTRKCNH2
SCHEMBL8609474 0.77 CCKBR (0.74) KCNH2CCKBRCCKAR
SCHEMBL8463081 0.77 KCNH2 (0.85) KCNH2CCKBR
SCHEMBL4421095 0.77 PSEN1 (0.82) OXTRKCNH2CCKBRNOTCH1RBPJ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776203-A4 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO INC (US) 1997-12-29 EP disclosed
EP-0776203-A1 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO. INC. (US) 1997-06-04 EP disclosed
US-5633251-A N-2,3-dihydro-1-(2-propyl)-2-oxo-5-phenyl-1h-1,4-benzodiazepines MERCK & CO., INC. (US) 1997-05-27 US disclosed
WO-1996005827-A1 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO., INC. (US) 1996-02-29 WO disclosed