SCHEMBL8760307

SCHEMBL8760307

CCCN1C(=O)C(NC(=O)Cc2cc(Cl)cc(Cl)c2)N=C(c2ccccc2)c2ccccc21

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.76
OXTR P30559 5/20 0.57
CCKBR P32239 11/20 0.55
NOTCH1 P46531 1/20 0.53
RBPJ Q06330 1/20 0.53
CCKAR P32238 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8760285 0.89 OXTR (0.64) KCNH2OXTRCCKBRNOTCH1RBPJ
SCHEMBL8461831 0.86 KCNH2 (1.00) KCNH2OXTR
SCHEMBL8462806 0.86 KCNH2 (1.00) KCNH2OXTR
SCHEMBL8760298 0.84 KCNH2 (0.69) KCNH2OXTRCCKBRCCKAR
SCHEMBL8761607 0.84 KCNH2 (0.69) KCNH2OXTRCCKBRCCKAR
SCHEMBL8761397 0.84 KCNH2 (0.69) KCNH2OXTRCCKBRCCKAR
SCHEMBL8745080 0.81 KCNH2 (0.89) KCNH2OXTR
SCHEMBL8852061 0.80 CCKBR (0.55) KCNH2CCKBRCCKAR
SCHEMBL4421095 0.80 PSEN1 (0.82) KCNH2OXTRCCKBRNOTCH1RBPJ
SCHEMBL8462635 0.80 KCNH2 (0.87) KCNH2OXTRCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776203-A4 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO INC (US) 1997-12-29 EP disclosed
EP-0776203-A1 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO. INC. (US) 1997-06-04 EP disclosed
WO-1996005827-A1 N-2,3-DIHYDRO-1-(2-PROPYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO., INC. (US) 1996-02-29 WO disclosed