SCHEMBL8760841

SCHEMBL8760841

NC(=O)c1ccc([N+](=O)[O-])c(N(CCCl)CCCl)c1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
CTSD P07339 1/20 0.36
CYP3A4 P08684 2/20 0.36
MAPT P10636 2/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
ALDH1A1 P00352 6/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
GAA P10253 1/20 0.33
PKM P14618 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
POLB P06746 2/20 0.33
PARP1 P09874 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CTDSP1 Q9GZU7 1/20 0.33
BCL2L1 Q07817 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2974936 0.79 TDP1 (0.35) KMT2ACYP3A4MAPTBLMPMP22
SCHEMBL8639690 0.78 SMN1; SMN2 (0.43) CYP3A4MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL8637449 0.76 ALDH1A1 (0.55) KMT2ACYP3A4MAPTBLMPMP22
SCHEMBL8635371 0.76 HCAR3 (0.39) CTSDMAPTALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL8633720 0.74 PARP1 (0.45) KMT2ACYP3A4MAPTALDH1A1LMNA
SCHEMBL5576910 0.74 LMNA (0.46) KMT2ACTSDCYP3A4MAPTBLM
SCHEMBL2364159 0.72 MAPT (0.47) KMT2ACTSDCYP3A4MAPTBLM
SCHEMBL29411996 0.72 MAPT (0.47) KMT2ACTSDCYP3A4MAPTBLM
SCHEMBL3421894 0.72 ALDH1A1 (0.50) KMT2ACYP3A4MAPTBLMPMP22
SCHEMBL667585 0.72 TSHR (0.54) KMT2ACYP3A4MAPTBLMPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0616609-B1 NITROANILINE DERIVATIVES AND THEIR USE AS ANTITUMOR AGENTS CANCER RES CAMPAIGN TECH (GB) 1997-06-18 EP disclosed
US-5571845-A Nitroaniline derivatives and their use as anti-tumour agents CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1996-11-05 US disclosed
WO-1993011099-A1 NITROANILINE DERIVATIVES AND THEIR USE AS ANTITUMOR AGENTS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1993-06-10 WO disclosed