SCHEMBL8761464

SCHEMBL8761464

FC(F)(F)c1nc(CCl)no1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MIF P14174 2/20 0.34
HDAC6 Q9UBN7 15/20 0.33
HDAC1 Q13547 8/20 0.33
HDAC8 Q9BY41 5/20 0.33
HDAC4 P56524 10/20 0.33
HDAC5 Q9UQL6 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9126570 0.83 MIF (0.33) MIFHDAC6HDAC1HDAC8HDAC4
SCHEMBL8761432 0.80 STAT3 (0.44)
SCHEMBL412107 0.80 HDAC6 (0.36) MIFHDAC6HDAC1HDAC8HDAC4
Hydrochloric Acid SCHEMBL439920 0.78 HDAC6 (0.35) MIFHDAC6HDAC1HDAC8HDAC4
SCHEMBL21634141 0.78 HDAC6 (0.34) MIFHDAC6HDAC1HDAC8HDAC4
SCHEMBL2308502 0.78 MIF (0.34) MIFHDAC6HDAC1HDAC8HDAC4
SCHEMBL478959 0.78 CNR2 (0.33)
SCHEMBL8233965 0.78 HDAC4 (0.39) MIFHDAC6HDAC1HDAC8HDAC4
SCHEMBL989859 0.77 HDAC6 (0.34) MIFHDAC6HDAC1HDAC8HDAC4
SCHEMBL13189194 0.75 MIF (0.35) MIFHDAC6HDAC1HDAC8HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250099448-A1 HETEROCYCLIC COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 2025-03-27 US disclosed
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed
CN-105940001-B Alternatively the new 7-azaindole derivatives of property histone deacetylase (HDAC) inhibitor and include its pharmaceutical composition 株式会社钟根堂 2018-02-06 CN disclosed
US-9650379-B2 Azaindole derivatives as selective histone deacetylase (HDAC) inhibitors and pharmaceutical compositions comprising the same CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2017-05-16 US disclosed
EP-3080125-A1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Chong Kun Dang Pharmaceutical Corp. (KR) 2016-10-19 EP disclosed
US-20160289230-A1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2016-10-06 US disclosed
WO-2015087151-A1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2015-06-18 WO disclosed
EP-0590415-B1 1,2,4-Oxadiazole derivatives for controlling endoparasites BAYER AG (DE) 1997-06-04 EP disclosed
US-5428047-A Nematocides BAYER AKTIENGESELLSCHAFT (DE) 1995-06-27 US disclosed
EP-0590415-A2 1,2,4-Oxadiazole derivatives for controlling endoparasites BAYER AG (DE) 1994-04-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250099448-A1 HETEROCYCLIC COMPOUNDS OPRM1, CYP1A1, CYP3A4 MIF 4268/4885HDAC6 634/4885HDAC1 271/4885
US-20160289230-A1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME HDAC5, HDAC1, HDAC2 MIF 1657/4885HDAC6 4/4885HDAC1 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.