SCHEMBL8762020

SCHEMBL8762020

Nc1cc(Cl)c(Cl)c(Cl)c1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
GAA P10253 1/20 0.40
DPP4 P27487 1/20 0.39
ALDH1A1 P00352 4/20 0.39
POLB P06746 1/20 0.39
TTR P02766 1/20 0.35
TSHR P16473 5/20 0.34
HSD17B10 Q99714 3/20 0.34
HPGD P15428 2/20 0.34
MAPK1 P28482 2/20 0.34
HSP90AA1 P07900 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
KDM4E B2RXH2 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
DAO P14920 2/20 0.33
TP53 P04637 1/20 0.33
TPMT P51580 1/20 0.33
CASP1 P29466 1/20 0.33
CD44 P16070 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10344814 0.83 CYP3A4 (0.48) CYP3A4GAADPP4ALDH1A1POLB
SCHEMBL8861080 0.82 KDM4E (0.40) CYP3A4GAADPP4ALDH1A1POLB
SCHEMBL11504756 0.79 CYP3A4 (0.48) CYP3A4DPP4ALDH1A1TTRTSHR
SCHEMBL7025073 0.77 ALDH1A1 (0.51) CYP3A4GAAALDH1A1TSHRHSD17B10
SCHEMBL8574199 0.76 GAA (0.47) GAAALDH1A1TSHRHSD17B10HPGD
SCHEMBL3136996 0.76 TSHR (0.43) CYP3A4DPP4ALDH1A1POLBTTR
SCHEMBL348918 0.74 CYP3A4 (0.53) CYP3A4GAADPP4ALDH1A1POLB
SCHEMBL7015064 0.74 DPP4 (0.48) CYP3A4DPP4ALDH1A1POLBTSHR
SCHEMBL31460347 0.74 THRB (0.44) CYP3A4GAADPP4ALDH1A1POLB
SCHEMBL2588215 0.74 DPP4 (0.46) CYP3A4DPP4ALDH1A1TTRTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107903269-A A kind of preparation method of three chlorine derivative of anagrelide 湖北省宏源药业科技股份有限公司 2018-04-13 CN claimed
CN-112142746-B Benzodiazepine compound, preparation method and medical application thereof 四川大学华西医院 2021-09-24 CN disclosed
CN-112142746-A Benzodiazepine compound, preparation method and medical application thereof 四川大学华西医院 2020-12-29 CN disclosed
CN-107903269-A A kind of preparation method of three chlorine derivative of anagrelide 湖北省宏源药业科技股份有限公司 2018-04-13 CN disclosed
EP-0781767-A1 Process for producing isatoic anhydrides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-07-02 EP disclosed