SCHEMBL8762111

SCHEMBL8762111

COC(=O)[C@H](CCSC)NCC1(Cc2ccccc2C)CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
GAA P10253 2/20 0.42
RECQL P46063 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
USP2 O75604 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TSHR P16473 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9015591 0.99 CYP3A4 (0.45) CYP3A4CYP2C19GAARECQLL3MBTL1
SCHEMBL8762105 0.82 CYP3A4 (0.50) CYP3A4CYP2C19GAARECQLL3MBTL1
SCHEMBL9015671 0.82 POLB (0.42) CYP3A4CYP2C19GAARECQLTSHR
Hydrochloric Acid SCHEMBL9015589 0.81 CYP3A4 (0.49) CYP3A4CYP2C19GAARECQLL3MBTL1
SCHEMBL8761068 0.72 CYP3A4 (0.36) CYP3A4CYP2C19GAARECQLUSP2
SCHEMBL1221538 0.69 LMNA (0.42) CYP3A4CYP2C19USP2ALDH1A1KDM4E
SCHEMBL1221603 0.69 ALDH1A1 (0.47) RECQLL3MBTL1ALDH1A1KDM4EKMT2A
SCHEMBL7848308 0.68 POLB (0.45) GAAL3MBTL1ALDH1A1KDM4EHTT
SCHEMBL27974457 0.68 USP2 (0.53) CYP3A4CYP2C19GAARECQLL3MBTL1
SCHEMBL2327387 0.68 USP2 (0.53) CYP3A4CYP2C19GAARECQLL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777475-A4 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 1997-12-03 EP disclosed
EP-0777475-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO. INC. (US) 1997-06-11 EP disclosed
WO-1996006609-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1996-03-07 WO disclosed