SCHEMBL9015671

SCHEMBL9015671

COC(=O)[C@H](CCSC)NCC1(Cc2ccccc2C)CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.42
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TSHR P16473 3/20 0.39
GPR119 Q8TDV5 2/20 0.38
YAP1 P46937 1/20 0.38
RECQL P46063 1/20 0.38
GAA P10253 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALOX15 P16050 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9015673 0.84 CYP3A4 (0.44) CYP3A4CYP2C19ALDH1A1TSHRYAP1
SCHEMBL8762111 0.82 CYP3A4 (0.45) POLBCYP3A4CYP2C19ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9015591 0.81 CYP3A4 (0.45) POLBCYP3A4CYP2C19ALDH1A1KDM4E
SCHEMBL7842738 0.78 POLB (0.45) POLBALDH1A1KDM4ETSHRGPR119
SCHEMBL7840954 0.77 POLB (0.53) POLBALDH1A1KDM4ETSHRMEN1
SCHEMBL7842880 0.73 PKM (0.52) POLBALDH1A1KDM4ETSHRKMT2A
SCHEMBL8762096 0.72 OPRD1 (0.44) POLBALDH1A1KDM4ETSHRGPR119
SCHEMBL8762050 0.71 GPR119 (0.44) POLBKDM4ETSHRGPR119KMT2A
SCHEMBL9015653 0.70 TSHR (0.42) POLBKDM4ETSHRGPR119ALOX15
SCHEMBL9015640 0.69 GPR119 (0.43) KDM4ETSHRGPR119ALOX15ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576313-A ENZYME INHIBITORS AND ANTICARCINOGENIC AGENTS MERCK & CO., INC. (US) 1996-11-19 US disclosed