SCHEMBL8763141

SCHEMBL8763141

CCCCOC(=O)NC(=O)[C@H](C)NC1CC(=O)OC1OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NAAA Q02083 4/20 0.42
CASP1 P29466 4/20 0.42
CASP3 P42574 4/20 0.42
CASP7 P55210 4/20 0.42
CASP6 P55212 4/20 0.42
CASP8 Q14790 4/20 0.42
CTSL P07711 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8763134 0.86 CASP1 (0.47) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL948901 0.85 KLK5 (0.43) CASP1CASP3CASP7CASP6CASP8
SCHEMBL948808 0.78 CASP3 (0.38) CASP1CASP3CASP7CASP6CASP8
SCHEMBL13776512 0.77 CASP3 (0.44) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL949530 0.76 CASP3 (0.38) CASP1CASP3CASP7CASP6CASP8
SCHEMBL950442 0.76 CASP3 (0.36) ALDH1A1CASP1CASP3CASP7CASP6
SCHEMBL12914558 0.76 CASP3 (0.48) CASP1CASP3CASP7CASP6CASP8
SCHEMBL948261 0.75 CASP3 (0.35) ALDH1A1CASP1CASP3CASP7CASP6
SCHEMBL949112 0.75 CASP1 (0.35) CASP1CASP3CASP7CASP6CASP8
SCHEMBL949260 0.75 NAAA (0.34) NAAACASP1CASP3CASP7CASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed