SCHEMBL8763145

SCHEMBL8763145

CC(=O)NCCC(CCc1ccncc1)C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
F13A1 P00488 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
MTNR1A P48039 2/20 0.41
MTNR1B P49286 1/20 0.41
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
TSHR P16473 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
ALDH1A1 P00352 2/20 0.38
ERAP2 Q6P179 2/20 0.38
ERAP1 Q9NZ08 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA5A P35218 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424305 0.78 KDM4E (0.65) KDM4EF13A1SMN1; SMN2RAB9ANPC1
SCHEMBL8763140 0.73 ACACB (0.43) SMN1; SMN2RAB9ANPC1TSHRLMNA
SCHEMBL8671157 0.73 KDM4E (0.53) KDM4EF13A1SMN1; SMN2RAB9ANPC1
SCHEMBL3055735 0.72 MTNR1A (0.55) MTNR1AMTNR1BANPEP
SCHEMBL3039933 0.72 MTNR1A (0.55) MTNR1AMTNR1BANPEP
SCHEMBL14795607 0.71 LOXL2 (0.45) SMN1; SMN2RAB9ANPC1HDAC2HDAC8
SCHEMBL18317154 0.69 HDAC2 (0.58) KDM4ESMN1; SMN2RAB9ANPC1HDAC2
Hydrochloric Acid SCHEMBL7204871 0.69 ERAP2 (0.51) SMN1; SMN2RAB9ALMNAERAP2ERAP1
Hydrochloric Acid SCHEMBL27556867 0.69 ERAP2 (0.51) SMN1; SMN2RAB9ALMNAERAP2ERAP1
SCHEMBL48578 0.68 HTT (0.64) SMN1; SMN2RAB9AHDAC6TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636141-B1 PYRIMIDINYL ACETAMIDES AS ELASTASE INHIBITORS ZENECA LTD (GB) 1997-06-25 EP disclosed