SCHEMBL8764336

SCHEMBL8764336

CNc1onc(C(F)(F)F)c1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.46
POLB P06746 2/20 0.42
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
BRD4 O60885 2/20 0.39
BRD2 P25440 1/20 0.39
MLYCD O95822 2/20 0.38
PTGS2 P35354 3/20 0.38
TSHR P16473 1/20 0.38
PTGS1 P23219 3/20 0.38
KDM4E B2RXH2 1/20 0.38
ENPP1 P22413 1/20 0.37
LMNA P02545 2/20 0.36
GLA P06280 1/20 0.36
MAT2A P31153 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27389289 0.76 BRD4 (0.61) TDO2BRD4BRD2PTGS2PTGS1
SCHEMBL9674379 0.75 PTGS1 (0.46) TDO2POLBESR1ESR2BRD4
SCHEMBL8764932 0.75 MLYCD (0.63) TDO2POLBESR1ESR2BRD4
SCHEMBL11014937 0.68 MLYCD (0.42) TDO2BRD4BRD2MLYCDPTGS2
SCHEMBL6151679 0.66 EDNRA (0.72) TSHR
SCHEMBL9063613 0.66 EDNRA (0.72) TSHR
SCHEMBL7849998 0.64 EDNRA (0.69) TSHR
SCHEMBL17532585 0.63 TDO2 (1.00) TDO2TSHRKDM4ETDP1
SCHEMBL5613767 0.62 EPHX2 (0.50) ESR1ESR2LMNA
SCHEMBL10503592 0.62 MLYCD (0.64) TDO2BRD4MLYCDENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375670-B1 Process for preparing 3-polyfluoroalkylisoxazolylamines SHIONOGI & CO (JP) 1997-08-06 EP disclosed
EP-0375670-A2 Process for preparing 3-polyfluoroalkylisoxazolylamines SHIONOGI & CO., LTD. (JP) 1990-06-27 EP disclosed