SCHEMBL876455

SCHEMBL876455

O=C(O)Oc1ccc2c(c1)C(=O)CC2

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.53
BRD4 O60885 1/20 0.50
HRH3 Q9Y5N1 2/20 0.48
MAOB P27338 5/20 0.46
MAOA P21397 4/20 0.46
GRM5 P41594 1/20 0.40
MAPK14 Q16539 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
BAZ1A Q9NRL2 1/20 0.37
MMP9 P14780 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688253 0.90 MAOA (0.57) PBRM1BRD4HRH3MAOBMAOA
SCHEMBL27819611 0.88 BRD4 (0.52) PBRM1BRD4HRH3MAOBMAOA
SCHEMBL10503926 0.81 PBRM1 (0.39) PBRM1BRD4HRH3MAOBMAOA
SCHEMBL3888850 0.81 RAB9A (0.53) PBRM1BRD4HRH3
Acetic Acid SCHEMBL6934641 0.80 MAOB (0.51) PBRM1BRD4HRH3MAOBMAPK14
SCHEMBL31638292 0.79 BRD4 (0.50) PBRM1BRD4HRH3MAOBMAOA
SCHEMBL10503520 0.79 PBRM1 (0.37) PBRM1BRD4HRH3MAOBMAOA
SCHEMBL8318501 0.79 MAOA (0.53) BRD4HRH3MAOBMAOAMAPK14
SCHEMBL10444174 0.78 KDM4E (0.45) GRM5MAPK14ALDH1A1MAPTSMN1; SMN2
SCHEMBL29243215 0.78 MAOA (0.55) PBRM1BRD4HRH3MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed