SCHEMBL8764606

SCHEMBL8764606

CS(=O)(=O)c1ccc(-c2c(-c3ccc(Cl)cc3Cl)c(C(F)(F)F)nn2-c2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.47
PTGS2 P35354 7/20 0.44
PTGS1 P23219 4/20 0.44
CNR2 P34972 3/20 0.41
CNR1 P21554 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766033 0.90 PTGS2 (0.55) OPRM1PTGS2PTGS1CNR2CNR1
SCHEMBL8765496 0.88 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL8765332 0.83 RXRA (0.49) PTGS2PTGS1CNR1
SCHEMBL8765403 0.78 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL8765194 0.78 PTGS2 (0.61) PTGS2PTGS1
SCHEMBL8765164 0.77 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8765317 0.77 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL8953746 0.76 RXRA (0.64) PTGS2PTGS1
SCHEMBL7778111 0.76 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL8654487 0.74 PTGS2 (0.57) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731794-B1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1997-08-06 EP disclosed
US-5639777-A 1,4,5-triphenyl pyrazolyl compounds for the treatment of inflammation and inflammation-related disorders G.D. SEARLE & CO. (US) 1997-06-17 US disclosed
US-5401765-A FOR TREATING ARTHRITIS, PAIN AND FEVER Searle, G. D. (US) 1995-03-28 US disclosed