SCHEMBL8764844

SCHEMBL8764844

CC(=O)NCCC1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
GRIN2B Q13224 11/20 0.57
CYP2C19 P33261 1/20 0.57
CYP2D6 P10635 4/20 0.56
CYP2C9 P11712 4/20 0.56
CYP3A4 P08684 3/20 0.53
FAAH O00519 1/20 0.53
TPSAB1 Q15661 2/20 0.52
TPSD1 Q9BZJ3 2/20 0.52
TPSG1 Q9NRR2 2/20 0.52
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19658451 0.93 SMN1; SMN2 (0.54) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL6654650 0.88 SMN1; SMN2 (0.62) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL16399970 0.86 HTT (0.56) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL7441282 0.85 TPSAB1 (0.56) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL15140566 0.85 SMN1; SMN2 (0.72) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL13519706 0.84 SMN1; SMN2 (0.67) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL27149310 0.83 SMN1; SMN2 (0.60) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL8765520 0.83 SMN1; SMN2 (0.62) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL13274303 0.83 HTT (0.69) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL1912329 0.83 KMT2A (0.57) HTTSMN1; SMN2NPC1RAB9AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625509-B1 N-alkyl substituted piperidine-derivatives with neurokinin receptor antagonist activity ZENECA LTD (GB) 1997-07-30 EP disclosed
US-5521199-A TREATMENT OF ASTHMA ZENECA LIMITED (GB) 1996-05-28 US disclosed
EP-0625509-A1 N-alkyl substituted piperidine-derivatives with neurokinin receptor antagonist activity ZENECA LIMITED (GB) 1994-11-23 EP disclosed