SCHEMBL8765170

SCHEMBL8765170

CS(=O)(=O)c1ccc(-c2cc(C(F)F)nn2-c2ccccc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.70
PTGS1 P23219 4/20 0.70
ALOX5 P09917 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002626 0.95 PTGS2 (0.77) PTGS2PTGS1ALOX5
SCHEMBL8954050 0.89 PTGS2 (0.65) PTGS2PTGS1
SCHEMBL8953911 0.89 PTGS2 (0.73) PTGS2PTGS1
SCHEMBL9003118 0.89 PTGS2 (0.73) PTGS2PTGS1
SCHEMBL8954509 0.89 PTGS2 (0.80) PTGS2PTGS1ALOX5
SCHEMBL9002971 0.88 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8635509 0.88 PTGS2 (0.78) PTGS2PTGS1
SCHEMBL9002995 0.88 PTGS2 (0.69) PTGS2PTGS1
SCHEMBL8953956 0.88 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8924564 0.88 PTGS2 (0.64) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731794-B1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1997-08-06 EP disclosed
US-5639777-A 1,4,5-triphenyl pyrazolyl compounds for the treatment of inflammation and inflammation-related disorders G.D. SEARLE & CO. (US) 1997-06-17 US disclosed
US-5401765-A FOR TREATING ARTHRITIS, PAIN AND FEVER Searle, G. D. (US) 1995-03-28 US disclosed