SCHEMBL8765272

SCHEMBL8765272

COc1ccc2c(c1)C[C@@H](OS(=O)(=O)c1ccc(C)cc1)CCC2

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.45
DRD2 P14416 5/20 0.45
DRD3 P35462 5/20 0.45
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
ACHE P22303 2/20 0.43
DRD4 P21917 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
HTR6 P50406 2/20 0.41
FKBP1A P62942 1/20 0.41
NAAA Q02083 1/20 0.39
ENPP3 O14638 1/20 0.39
ENPP1 P22413 1/20 0.39
ENPP2 Q13822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765278 1.00 CYP2D6 (0.45) CYP2D6DRD2DRD3CA1CA2
SCHEMBL8766442 1.00 CYP2D6 (0.45) CYP2D6DRD2DRD3CA1CA2
SCHEMBL6401807 0.93 DRD2 (0.50) CYP2D6DRD2DRD3CA1CA2
SCHEMBL8766020 0.82 DRD2 (0.51) DRD2DRD3CA1CA2ACHE
SCHEMBL9630809 0.77 CYP19A1 (0.52) DRD2DRD3CA1CA2ACHE
SCHEMBL6198029 0.74 CYP2D6 (0.63) CYP2D6CA1CA2ACHEALDH1A1
SCHEMBL6198035 0.74 CYP2D6 (0.63) CYP2D6CA1CA2ACHEALDH1A1
SCHEMBL777214 0.74 CYP2D6 (0.63) CYP2D6CA1CA2ACHEALDH1A1
SCHEMBL2670048 0.74 CYP2D6 (0.63) CYP2D6CA1CA2ACHEALDH1A1
SCHEMBL6405616 0.74 DRD2 (0.57) DRD2DRD3CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0583485-B1 ETHANOLAMINE DERIVATIVES HAVING SYMPATHOMIMETIC AND ANTI-POLLAKIURIA ACTIVITIES FUJISAWA PHARMACEUTICAL CO (JP) 1997-08-13 EP disclosed
US-5387710-A Ethanolamine derivatives having sympathomimetic and anti-pollakiuria activities FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-02-07 US disclosed
EP-0583485-A1 ETHANOLAMINE DERIVATIVES HAVING SYMPATHOMIMETIC AND ANTI-POLLAKIURIA ACTIVITIES. FUJISAWA PHARMACEUTICAL CO (JP) 1994-02-23 EP disclosed
WO-1993015041-A1 ETHANOLAMINE DERIVATIVES HAVING SYMPATHOMIMETIC AND ANTI-POLLAKIURIA ACTIVITIES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-08-05 WO disclosed