SCHEMBL8765441

SCHEMBL8765441

C[Si](C)(C)C#CC1CCc2ccccc2S1

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.35
PDPK1 O15530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141643 0.75 SIGMAR1 (0.39) SIGMAR1PDPK1
SCHEMBL30715562 0.75 SIGMAR1 (0.39) SIGMAR1PDPK1
SCHEMBL7783911 0.75 SIGMAR1 (0.39) SIGMAR1
SCHEMBL6666465 0.75 SIGMAR1 (0.39) SIGMAR1PDPK1
SCHEMBL9765060 0.71 SIGMAR1 (0.38) SIGMAR1
SCHEMBL9125425 0.69 PLAU (0.43)
SCHEMBL30724832 0.69 SIGMAR1 (0.42) SIGMAR1PDPK1
SCHEMBL10780065 0.69 SIGMAR1 (0.42) SIGMAR1PDPK1
SCHEMBL6721448 0.66 SIGMAR1 (0.43) SIGMAR1PDPK1
SCHEMBL16340795 0.66 TSHR (0.35) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1997-07-30 EP disclosed
WO-1996011686-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-04-25 WO disclosed
EP-0419132-A2 Process and intermediates for preparing compounds having a disubstituted acetylene moiety and retinoic acid-like biological activity ALLERGAN, INC. (US) 1991-03-27 EP disclosed