SCHEMBL8766148

SCHEMBL8766148

CCOP(=O)(OCC)C(c1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1)N(CCCc1ccccc1)C(C)=O

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 3/20 0.46
LMNA P02545 3/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
GAA P10253 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NR1I2 O75469 1/20 0.36
POLB P06746 1/20 0.36
FDPS P14324 2/20 0.36
RECQL P46063 1/20 0.36
FDFT1 P37268 1/20 0.35
TACR1 P25103 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766484 0.93 HMGCR (0.38) HMGCRLMNAGAAMEN1KMT2A
SCHEMBL8766996 0.91 HMGCR (0.44) HMGCRLMNAALDH1A1MAPTGAA
SCHEMBL8766505 0.90 MEN1 (0.39) HMGCRLMNAGAAMEN1KMT2A
SCHEMBL8766187 0.89 HMGCR (0.46) HMGCRLMNAGAAMEN1KMT2A
SCHEMBL8766605 0.87 FDPS (0.41) LMNAGAAMEN1KMT2AFDPS
SCHEMBL8766091 0.87 HMGCR (0.41) HMGCRLMNAALDH1A1MAPTGAA
SCHEMBL8766586 0.82 MEN1 (0.43) HMGCRLMNAALDH1A1MAPTGAA
SCHEMBL7128247 0.78 HMGCR (0.47) HMGCRLMNAALDH1A1MAPTGAA
SCHEMBL8766613 0.76 HMGCR (0.49) HMGCRMAPTGAAMEN1KMT2A
SCHEMBL7119208 0.74 HMGCR (0.43) HMGCRLMNAGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559079-B1 Substituted aminophosphonate derivatives, process for their preparation and pharmaceutical compositions containing them SYMPHAR SA (CH) 1997-08-13 EP claimed
EP-0559079-A1 Substituted aminophosphonate derivatives, process for their preparation and pharmaceutical compositions containing them SYMPHAR S.A. (CH) 1993-09-08 EP claimed
EP-0559079-B1 Substituted aminophosphonate derivatives, process for their preparation and pharmaceutical compositions containing them SYMPHAR SA (CH) 1997-08-13 EP disclosed
US-5424303-A For treating hypercholesterolemia and hyperlipidemia SYMPHAR SA (CH) 1995-06-13 US disclosed
EP-0559079-A1 Substituted aminophosphonate derivatives, process for their preparation and pharmaceutical compositions containing them SYMPHAR S.A. (CH) 1993-09-08 EP disclosed