SCHEMBL8766182

SCHEMBL8766182

CCOP(=O)(OCC)C(Nc1ccc(N2C(=O)c3ccc(Cl)cc3C2=O)c(C)c1)c1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ERBB2 P04626 1/20 0.39
NPSR1 Q6W5P4 2/20 0.38
GRM1 Q13255 5/20 0.38
GRM4 Q14833 5/20 0.38
HMGCR P04035 1/20 0.38
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
LMNA P02545 4/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.35
GAA P10253 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973534 0.81 CA12 (0.56) CA12CA1CA2CA9L3MBTL1
SCHEMBL8766495 0.76 ESR1 (0.37) CA12CA1CA2CA9ERBB2
SCHEMBL8766175 0.72 CA12 (0.57) CA12CA1CA2CA9NPSR1
SCHEMBL8767390 0.71 ESR1 (0.40) ERBB2GRM1GRM4ESR1ESR2
SCHEMBL14560075 0.71 ERBB2 (0.51) ERBB2GRM1GRM4ESR1ESR2
SCHEMBL7119145 0.68 HMGCR (0.46) L3MBTL1NPSR1HMGCRLMNAMAPT
SCHEMBL11787416 0.67 GRM1 (0.53) CA12CA1CA9ERBB2GRM1
SCHEMBL5903417 0.67 ESR1 (0.61) ERBB2GRM1GRM4ESR1ESR2
SCHEMBL9403099 0.64 HMGCR (0.45) CA12CA1CA2CA9NPSR1
SCHEMBL13222267 0.64 ERBB2 (0.51) ERBB2GRM1GRM4ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559079-B1 Substituted aminophosphonate derivatives, process for their preparation and pharmaceutical compositions containing them SYMPHAR SA (CH) 1997-08-13 EP claimed
EP-0559079-A1 Substituted aminophosphonate derivatives, process for their preparation and pharmaceutical compositions containing them SYMPHAR S.A. (CH) 1993-09-08 EP claimed