SCHEMBL8767390

SCHEMBL8767390

Cc1cc(N(CP(=O)(O)O)c2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)ccc1N1C(=O)c2ccc(Cl)cc2C1=O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
GRM1 Q13255 13/20 0.37
GRM4 Q14833 9/20 0.37
ERBB2 P04626 1/20 0.35
CYP1A2 P05177 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
GAA P10253 1/20 0.32
POLB P06746 1/20 0.31
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766495 0.89 ESR1 (0.37) ESR1ESR2GRM1GRM4ERBB2
SCHEMBL8766469 0.78 LMNA (0.38) CYP1A2MEN1KMT2AGAAPOLB
SCHEMBL8766182 0.71 CA12 (0.39) ESR1ESR2GRM1GRM4ERBB2
SCHEMBL8766028 0.71 LMNA (0.40) CYP1A2MEN1KMT2AGAAPOLB
SCHEMBL5903417 0.70 ESR1 (0.61) ESR1ESR2GRM1GRM4ERBB2
SCHEMBL8766961 0.69 GAA (0.39) MEN1KMT2AGAAPOLBLMNA
SCHEMBL8766614 0.68 GAA (0.49) CYP1A2MEN1KMT2AGAAPOLB
SCHEMBL8766637 0.67 CA1 (0.46) MEN1KMT2AGAALMNA
SCHEMBL8766723 0.65 HMGCR (0.39) MEN1KMT2AGAALMNA
SCHEMBL5903671 0.65 ESR1 (0.54) ESR1ESR2GRM1GRM4ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559079-B1 Substituted aminophosphonate derivatives, process for their preparation and pharmaceutical compositions containing them SYMPHAR SA (CH) 1997-08-13 EP claimed