SCHEMBL8767150

SCHEMBL8767150

CCOc1ccc(-c2cc(F)c(C#Cc3ccc(F)c(F)c3)c(F)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.41
FFAR4 Q5NUL3 2/20 0.39
FFAR1 O14842 1/20 0.39
NQO1 P15559 1/20 0.39
ERN1 O75460 1/20 0.38
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MCHR1 Q99705 2/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CHRM1 P11229 1/20 0.36
HTR2A P28223 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766249 0.90 RARA (0.41) ERN1MCHR1CHRM1HTR2AGRM5
SCHEMBL8767188 0.89 RARB (0.45) FFAR4FFAR1ERN1ALDH1A1NPC1
SCHEMBL9469188 0.85 NQO1 (0.50) NQO1ALDH1A1GRM5CACNA1C
SCHEMBL8767592 0.85 CHRNA7 (0.40) CHRNA7NQO1CYP11B1CYP11B2ALDH1A1
SCHEMBL9433084 0.84 CHRNA7 (0.39) CHRNA7NQO1CYP11B1CYP11B2ALDH1A1
SCHEMBL9433854 0.84 MAOB (0.38) ALDH1A1MCHR1MAPTSMN1; SMN2CHRM1
SCHEMBL8766246 0.83 CYP17A1 (0.39) CYP11B1CYP11B2L3MBTL1GRM5
SCHEMBL9751747 0.82 NQO1 (0.54) CHRNA7FFAR4FFAR1NQO1CYP11B1
SCHEMBL8766258 0.81 CYP17A1 (0.37) CYP11B1CYP11B2ALDH1A1NPC1RAB9A
SCHEMBL9434250 0.79 MCHR1 (0.40) ERN1NPC1RAB9AMCHR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543244-B1 Fluoro substituted tolans and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 1997-08-20 EP disclosed
US-5372746-A Fluoro-substituted tolane compounds and liquid crystalline mixtures containing same HOFFMANN-LA ROCHE INC. (US) 1994-12-13 US disclosed
EP-0543244-A1 Fluoro substituted tolans and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed