SCHEMBL8767333

SCHEMBL8767333

Nc1ccnn1-c1c(Cl)cc(C(F)F)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
KDR P35968 2/20 0.36
KDM4E B2RXH2 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
RIPK2 O43353 1/20 0.32
EGFR P00533 1/20 0.32
SRC P12931 1/20 0.32
BRAF P15056 1/20 0.32
TNK2 Q07912 1/20 0.32
PTK6 Q13882 1/20 0.32
MINK1 Q8N4C8 1/20 0.32
GABRA2 P47869 2/20 0.32
GABRB2 P47870 2/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9459015 0.81 KDR (0.51) POLBKDRKDM4ERIPK2EGFR
SCHEMBL10496963 0.80 POLB (0.37) POLBKDRKDM4E
SCHEMBL9458856 0.77 GABRB3 (0.54) GABRA2GABRB2GABRPGABRDGABRA1
SCHEMBL17844034 0.75 POLB (0.52) POLBKDRKDM4E
SCHEMBL7082414 0.74 MAPT (0.41) POLBKDRKDM4EGABRA2GABRB2
SCHEMBL9822871 0.71 POLB (0.37) POLBKDRKDM4EGABRA2GABRB2
SCHEMBL8767317 0.69 L3MBTL1 (0.49) KDM4ETRPV4
SCHEMBL10389922 0.69 POLB (0.35) POLBKDRGABRA2GABRB2GABRP
SCHEMBL7086689 0.69 GABRB3 (0.45) GABRA2GABRB2GABRPGABRDGABRA1
SCHEMBL1727194 0.68 POLB (0.47) POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0788484-A1 2-CHLORO-N- 1-(2,6-DICHLORO-4-DIFLUOROMETHYL-PHENYL)-1H-PYRAZOL-5-YL]-PROPANAMIDE AND A METHOD OF PRODUCING THE SAME BAYER AG (DE) 1997-08-13 EP claimed
WO-1996012707-A1 2-CHLORO-N-[1-(2,6-DICHLORO-4-DIFLUOROMETHYL-PHENYL)-1H-PYRAZOL-5-YL]-PROPANAMIDE AND A METHOD OF PRODUCING THE SAME BAYER AKTIENGESELLSCHAFT (DE) 1996-05-02 WO claimed
JP-1066170-A None JP disclosed
EP-0788484-A1 2-CHLORO-N- 1-(2,6-DICHLORO-4-DIFLUOROMETHYL-PHENYL)-1H-PYRAZOL-5-YL]-PROPANAMIDE AND A METHOD OF PRODUCING THE SAME BAYER AG (DE) 1997-08-13 EP disclosed
WO-1996012707-A1 2-CHLORO-N-[1-(2,6-DICHLORO-4-DIFLUOROMETHYL-PHENYL)-1H-PYRAZOL-5-YL]-PROPANAMIDE AND A METHOD OF PRODUCING THE SAME BAYER AKTIENGESELLSCHAFT (DE) 1996-05-02 WO disclosed
EP-0303906-A1 1-Aryl pyrazoles BAYER AG (DE) 1989-02-22 EP disclosed
EP-0303153-A2 1-Aryl pyrazoles BAYER AG (DE) 1989-02-15 EP disclosed