SCHEMBL8768166

SCHEMBL8768166

CCCCCCCN(Cc1ccc(OCCCCC(=O)OCC)cc1)C(=O)Nc1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 2/20 0.52
CNR2 P34972 1/20 0.48
HDAC1 Q13547 3/20 0.46
PTGES O14684 1/20 0.45
LTA4H P09960 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HDAC6 Q9UBN7 3/20 0.43
HDAC3 O15379 2/20 0.43
HDAC4 P56524 2/20 0.43
HDAC7 Q8WUI4 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
HDAC9 Q9UKV0 2/20 0.43
HDAC5 Q9UQL6 2/20 0.43
HRH3 Q9Y5N1 1/20 0.43
PPARG P37231 1/20 0.43
PPARD Q03181 1/20 0.43
PPARA Q07869 1/20 0.43
EPHX2 P34913 1/20 0.43
HDAC10 Q969S8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9258955 0.85 CNR2 (0.53) CCKBRCNR2HDAC1PTGESLTA4H
SCHEMBL9260018 0.81 HDAC6 (0.47) CNR2HDAC1PTGESHDAC6HDAC3
SCHEMBL8767865 0.81 SOAT1 (0.64) HRH3PPARGPPARDPPARA
SCHEMBL8768869 0.81 PPARA (0.56) CCKBRCNR2HDAC1HDAC6HDAC3
SCHEMBL8768812 0.81 PPARA (0.56) CCKBRCNR2HDAC1HDAC6HDAC3
SCHEMBL9784546 0.78 SOAT1 (0.50) CNR2HDAC1ALDH1A1HDAC6HDAC3
SCHEMBL8768663 0.77 PPARA (0.69) CNR2HDAC1ALDH1A1HDAC6HDAC3
SCHEMBL13018713 0.77 HDAC6 (0.67) CNR2HDAC1ALDH1A1HDAC6HDAC3
SCHEMBL9784419 0.77 THRB (0.47) CNR2HDAC1HDAC6
SCHEMBL10888065 0.76 HDAC6 (0.63) HDAC1ALDH1A1HDAC6HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639178-B1 ANTI-ATHEROSCLEROTIC ARYL COMPOUNDS WELLCOME FOUND (GB) 1997-09-03 EP disclosed
US-5658944-A ANTICHOLESTEROL AGENTS THE UNIVERSITY OF SOUTH CAROLINA (US) 1997-08-19 US disclosed