SCHEMBL8768882

SCHEMBL8768882

Cc1cc(C#N)ccc1Nc1c(NCCc2ccccc2)c(=O)c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 4/20 0.50
CCNC P24863 2/20 0.46
CDK8 P49336 2/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
CTDSP1 Q9GZU7 1/20 0.46
CDKN1A P38936 1/20 0.44
CDK19 Q9BWU1 1/20 0.44
ABCC9 O60706 1/20 0.42
ABCC8 Q09428 1/20 0.42
KCNJ11 Q14654 1/20 0.42
KCNJ8 Q15842 1/20 0.42
POLB P06746 1/20 0.41
HDAC1 Q13547 1/20 0.41
FES P07332 1/20 0.41
FGFR1 P11362 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41
TAAR1 Q96RJ0 2/20 0.39
ALDH1A1 P00352 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8768922 0.79 CXCR2 (0.50) CXCR2CCNCCDK8MEN1KMT2A
SCHEMBL8870610 0.76 ABCC9 (0.53) CXCR2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8870608 0.76 ABCC9 (0.53) CXCR2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8768157 0.74 CXCR2 (0.45) CXCR2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8768613 0.73 GSK3B (0.50) CXCR2MEN1KMT2ACTDSP1HDAC1
SCHEMBL8768944 0.72 GAA (0.50) CXCR2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL19956899 0.70 MEN1 (0.63) CXCR2MEN1KMT2ACTDSP1POLB
SCHEMBL30673020 0.69 CNR1 (0.46) CXCR2MEN1KMT2AHDAC1FES
SCHEMBL5765787 0.69 CCNC (0.57) CCNCCDK8CDKN1ACDK19POLB
SCHEMBL8768997 0.68 CXCR2 (0.42) CXCR2CCNCCDK8MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0789690-A1 N-ARYL AND N-HETEROARYL-1,2-DIAMINOCYCLOBUTENE-3,4-DIONES WITH SMOOTH MUSCLE RELAXING ACTIVITIES AMERICAN HOME PRODUCTS CORPORATION (US) 1997-08-20 EP claimed
WO-1996014300-A1 N-ARYL AND N-HETEROARYL-1,2-DIAMINOCYCLOBUTENE-3,4-DIONES WITH SMOOTH MUSCLE RELAXING ACTIVITIES AMERICAN HOME PRODUCTS CORPORATION (US) 1996-05-17 WO claimed