SCHEMBL8768922

SCHEMBL8768922

N#Cc1cccc(Nc2c(NCCc3ccccc3)c(=O)c2=O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 4/20 0.50
LMNA P02545 1/20 0.49
FLT4 P35916 2/20 0.48
KDR P35968 2/20 0.48
FES P07332 1/20 0.48
FGFR1 P11362 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
CCNC P24863 2/20 0.44
CDK8 P49336 2/20 0.44
CDKN1A P38936 1/20 0.44
CDK19 Q9BWU1 1/20 0.44
CTDSP1 Q9GZU7 1/20 0.43
KCNA5 P22460 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPKAPK2 P49137 1/20 0.42
FLT1 P17948 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 1/20 0.42
HDAC1 Q13547 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8768882 0.79 CXCR2 (0.50) CXCR2FLT4KDRFESFGFR1
SCHEMBL8349873 0.78 L3MBTL1 (0.58) LMNACCNCCDK8CDKN1ACDK19
SCHEMBL30673020 0.77 CNR1 (0.46) CXCR2FLT4KDRFESFGFR1
SCHEMBL4364173 0.74 FLT4 (0.79) CXCR2FLT4KDRFESFGFR1
SCHEMBL30673004 0.74 MEN1 (0.62) CXCR2LMNAFLT4KDRFES
SCHEMBL30513604 0.74 GRM4 (0.48) CXCR2LMNAFLT4KDRMAPKAPK2
SCHEMBL28652875 0.74 GRM4 (0.48) CXCR2LMNAFLT4KDRMAPKAPK2
SCHEMBL4370740 0.73 FLT4 (0.56) CXCR2FLT4KDRFESFGFR1
SCHEMBL4366404 0.73 FES (0.56) CXCR2FLT4KDRFESFGFR1
SCHEMBL8868951 0.73 MAPKAPK2 (0.59) CXCR2MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0789690-A1 N-ARYL AND N-HETEROARYL-1,2-DIAMINOCYCLOBUTENE-3,4-DIONES WITH SMOOTH MUSCLE RELAXING ACTIVITIES AMERICAN HOME PRODUCTS CORPORATION (US) 1997-08-20 EP disclosed
WO-1996014300-A1 N-ARYL AND N-HETEROARYL-1,2-DIAMINOCYCLOBUTENE-3,4-DIONES WITH SMOOTH MUSCLE RELAXING ACTIVITIES AMERICAN HOME PRODUCTS CORPORATION (US) 1996-05-17 WO disclosed